Papers of Krzysztof Wojciechowski
1978-1988  1989-1993  1994-1999  2000-2002    2003-  
Institute of Organic Chemistry


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Scientific activities
  1. M. Mąkosza, K. Wojciechowski, M. Jawdosiuk "Aromatic Nucleophilic Substitution in Chloronitrobenzenes by Carbanions Derived from N-­Substituted Oxindoles" Pol. J. Chem. 1978, 52, 1173.
  2. M. Fedoryński, K. Wojciechowski, Z. Matacz, M. Mąkosza "Sodium and Potassium Carbonates: Efficient Strong Bases in Solid-liquid Two-Phase Systems" J. Org. Chem. 1978, 43, 4682.
  3. M. Jawdosiuk, A. Jończyk, A. Kwast, M. Mąkosza, I. Kmiotek-­Skarżyńska, K. Wojciechowski "9-­Chlorofluorene Transformations in Catalytic Two­Phase Systems"  Pol. J. Chem. 1979, 53, 191.
  4. L. Ghosez, J.­P. Antoine, E. Deffense, M. Navarro, V. Libert, M. J. O'Donnell, W. A. Bruder, K. Willey, K. Wojciechowski "Synthesis of Amino Acids. Alkylation of Aldimine and Ketimine Derivatives of Glycine Ethyl Ester under Various Phase-Ttransfer Conditions"  Tetrahedron Lett. 1982, 23, 4255.
  5. M. J. O'Donnell, K. Wojciechowski, L. Ghosez, M. Navarro, F. Sainte, J.­P. Antoine "Alkylation of Protected ­Amino Acids in the Presence of Potassium Carbonate"  Synthesis 1984, 313.
  6. M. J. O'Donnell, W. A. Bruder, B. W. Daugherty, D. Liu, K. Wojciechowski, "Nitrogen Alkylation of Schiff Bases and Amidines as a Route to N-­Alkyl Amino Acids"  Tetrahedron Lett. 1984, 25, 651.
  7. M. Mąkosza, K. Wojciechowski, "Intramolecular Vicarious Nucleophilic Substitution of Hydrogen"  Tetrahedron Lett. 1984, 25, 4791.
  8. K. Wojciechowski, M. Mąkosza, "New Synthesis of Indole Derivatives via Vicarious Nucleophilic Substitution of Hydrogen"  Tetrahedron Lett. 1984, 25, 4793.
  9. M. Mąkosza, K. Wojciechowski, "Synthesis of Phosphonic Acid Esters in Solid-­Liquid Two­Phase System"  Bull. Pol. Acad. Sci. Chemistry  1984, 32, 175.
  10. K. Wojciechowski, M. Mąkosza, "Synthesis of 2-­Arylindoles via Condensation of ortho­Aminobenzyl Sulfones with Aromatic Aldehydes" Bull. Soc. Chim. Belg. 1986, 95, 671.
  11. K. Wojciechowski, M. Mąkosza, "A Facile Synthesis of 3-Sulfonyl Substituted Indole Derivatives" Synthesis 1986, 651.
  12. M. Mąkosza, W. Danikiewicz, K. Wojciechowski, "Reactions of ­Chloroalkyl Sulfones with Nitronaphthalene Derivatives" Liebigs Ann. Chem. 1987, 711.
  13. M. Mąkosza, W. Danikiewicz, K. Wojciechowski, "Simple and General Synthesis of Hydroxy­ and Methoxyindoles via Vicarious Nucleophilic Substitution of Hydrogen" Liebigs Ann. Chem. 1988, 203.
  14. K. Wojciechowski, "Efficient Synthesis of alpha-­Chlorovinyl Phenyl Sulfone" Org. Prep. Proc. Intl. 1988, 20, 493.
  15. K. Wojciechowski, "Reactions of Fluorene Derivatives Carbanions with Aromatic Nitro Compounds" Bull. Pol. Acad. Sci. Chemistry 1988, 36, 235..
  16. K. Wojciechowski, W. Danikiewicz, M. Mąkosza, "Synthesis of Hydroxyindoles via Vicarious Nucleophilic Substitution" in Chemistry of Heterocyclic Compounds Studies in Organic Chemistry 35, (J. Kovac and P. Zalupsky, Eds.), Elsevier, Amsterdam 1988. 
  17. K. Wojciechowski, M. Mąkosza, "Vicarious Nucleophilic Substitution in 5- ­and 6-­Nitroindole Derivatives" Synthesis 1989, 106.
  18. M. Mąkosza, W. Danikiewicz, K. Wojciechowski, "Vicarious Nucleophilic Substitution with Sulfur Containing Carbanions" Phosphorus, Sulfur, and Silicon 1990, 53, 457. (Review)
  19. M. Mąkosza, K. Sienkiewicz, K. Wojciechowski, "Vicarious Nucleophilic Substitution of Hydrogen in Nitroarenes by Carbanions of Alkyl Dichloroacetates. Some New Transformations of Chloro(nitroaryl)acetates" Synthesis 1990, 850.
  20. S. Ostrowski, K. Wojciechowski, "Vicarious Nucleophilic Substitution of Hydrogen in Nitrobenzofuroxanes and the Boulton-­Katritzky Rearrangement of the VNS products" Can. J. Chem. 1990, 68, 2239.
  21. K. Wojciechowski, "Synthesis of 4-Nitro-2H-isoindole Derivatives" Liebigs.Ann. Chem. 1991, 831.
  22. K. Wojciechowski "Synthesis of 1,2,3,4-Tetrahydroquinoline-2,3-dicarboxylic Acid Derivatives" Synlett 1991, 571.
  23. K. Wojciechowski, M. Mąkosza "Synthesis of Benzosultams via intramolecular Vicarious Nucleophilic Substitution of Hydrogen" Synthesis 1992, 571.
  24. K. Wojciechowski "Synthesis of 2,1-Benzisothiazoline 2,2-Dioxide Derivatives" Pol. J. Chem. 1992, 66, 1121.
  25. Z. Wróbel, K. Wojciechowski "Nitroarylation of Nitrobenzyl Derivatives" Pol. J. Chem. 1992, 66, 1125.
  26. K. Wojciechowski "Reactions of Aza-ortho-xylylenes Generated from 2,1-Benzisothiazoline 2,2-Dioxides" Tetrahedron 1993, 49, 7277.
  27. K. Wojciechowski "New Synthesis of 2-Phenylindene Derivatives" Synth. Commun. 1993, 23, 2415.
  28. W. Danikiewicz, K. Wojciechowski, R.H. Fokkens, N.M.M. Nibbering "Electron Impact-induced Fragmentation of 2,1-Benzisothiazoline 2,2-Dioxides" Org. Mass Spectrom. 1993, 28, 853.
  29. K. Wojciechowski "[1,5] Hydrogen Shift in Aza-ortho-xylylenes Generated from 3-Alkyl-2,1-benzisothiazoline 2,2-Dioxides" Tetrahedron 1993, 49, 10017.
  30. W. Danikiewicz, K. Wojciechowski, R.H. Fokkens, N.M.M. Nibbering "On the Mechanisms of Electron-impact-induced Sulfur Dioxide Elimination from the Molecular Ions of 4-Nitro- and 6-Nitro-2,1-benzisothiazoline 2,2-Dioxide Derivatives" Rapid Commun. Mass Spectrom. 1993, 7, 763. 
  31. K. Mąkosza, R. Kuciak, K. Wojciechowski "Vicarious Nucleophilic Substitution of Hydrogen in Azulenes" Liebigs Ann. Chem. 1994, 615.
  32. W. Danikiewicz, K.Wojciechowski, M.Olejnik "Generation and Reactions of Aza-ortho-xylylenes in the Injector of GC/MS System" Tetrahedron Lett. 1995, 36, 1099.
  33. W. Danikiewicz, K. Wojciechowski "Alkyl Group Migration during Fragmentation of N-(alkoxymethyl)sulfonamides Following Electron Ionization" Rapid Commun. Mass Spectrom. 1996, 10, 763.
  34. K Wojciechowski "Transformations of Cumulated Aza-ortho-xylylenes Generated from 3-Arylmethylene-2,1-benzisothiazoline 2,2-Dioxides" Molecules 1996, 1, 51-56.
  35. K Wojciechowski "Synthesis of Nitrobenzophenones from Nitro--sulfonyldiphenylmethane Derivatives", Synth.Commun. 1997, 26, 135-144.
  36. M. Mąkosza, J. Stalewski, K. Wojciechowski, W. Danikiewicz "Synthesis of 1,3,4,5-Tetrahydrobenz[cd]indole via the Vicarious Nucleophilic Substitution of Hydrogen", Tetrahedron, 1997, 53, 193-214.
  37. W. Danikiewicz, K. Wojciechowski "Fragmentation of 1-alkyl derivatives of 5- and 7-nitro-2,1-benzisothiazoline 2,2-dioxides upon electron ionization" Eur. Mass. Spectrom. 1997, 3, 55-65
  38. M. Mąkosza, K. Wojciechowski "Applications of Vicarious Nucleophilic Substitution in Organic Synthesis" Liebigs Ann. Chem. 1997, 1805-1816 (Review).
  39. K. Wojciechowski, Sz. Kosiński "Genaration and Reactions of Heteroanalogues of Aza-ortho-xylylenes" Tetrahedron Lett. 1997, 38, 4667-4670.
  40. K. Wojciechowski "Generation and Reactions of Aza-ortho-xylylenes" Pol. J. Chem. 1997, 71, 1375-1400 (Review).
  41. W. Danikiewicz, K. Wojciechowski "Fragmentation of 1-Methyl-1,2,3,4-tetrahydroquinoline-2,3-dicarboxylic Acid Derivaitves upon Electron Ionisation" Pol. J. Chem. 1998, 72, 554-563.
  42. Sz. Kosiński, K. Wojciechowski "Reactions of Aza-ortho-xylylenes with 1,4-Naphthoquinone" Pol. J. Chem. 1998, 72, 2546-2550.
  43. W. Danikiewicz, K. Wojciechowski  "Fragmentation of ionized N-(alkoxymethyl)sulfon-amides: An Alkyl Group Migration", in: "Fundamentals and Applications of Gas Phase Ion Chemistry" Ed. K.R. Jennings, s. 406, Kluwer Academic Publishers, Dordrecht 1999.
  44. A. Chrostowska, F. Gracian, J.-M. Sotiropoulos, G. Pfister-Guillouzo, K. Wojciechowski "Application of Photoelectron Spectroscopy to Molecular Properties, 57. UV photoelectron Spectroscopy Studies of the Products of Thermal Extrusion of Sulfur Dioxide from Benzosultams" Eur. J. Org. Chem. 2000, 313-318.
  45. S. Kosiński, K. Wojciechowski "Reactions of Heteroanalogues of Aza-ortho-xylylenes generated from 1,3-dialkylpyridosultams" Eur. J. Org. Chem. 2000, 1263-1270.
  46. M. Mąkosza, K. Wojciechowski "Nucleophilic Aromatic Substitution of Hydrogen as a Tool for the Synthesis of Indole and Quinoline Derivatives" Heterocycles 2001, 54, 445-474 (Review)
  47. W. Danikiewicz, K. Wojciechowski, S. Kosiński, M. Olejnik, "EI-Induced Fragmentation of 3-Cyclopropanospiro and 3-Cyclobutanospiro Derivatives of Benzo- and Pyridosultams"  J. Mass Spectrom. 2001, 36, 430-440.
  48. K. Wojciechowski, S. Kosiński "Synthesis of Novel Isothiazolo[4,3-b]-pyridine and Isothiazolo[4,3-b]quinoline Derivatives" Tetrahedron 2001, 57, 5009-5014.
  49. M. Mąkosza, M. Barbasiewicz, K. Wojciechowski "Can nitroalkanes be obtained directly from alcohols and sodium nitrite in acetic acid - hydrochloric acid mixture?" Synlett 2001, 1121-1122.
  50. K. Wojciechowski "Aza-ortho-xylylenes in Organic Synthesis" Eur. J. Org. Chem. 2001, 3587-3605 (Review)
  51. K. Wojciechowski, S. Kosiński "Reactions of Pyridine Analogues of Aza-ortho-xylylenes Generated from 1,3-Dihydroisothiazolo[4,3-b]pyridine 2,2-Dioxides (Pyridosultams). Formation of 2:1 Adducts with N-Phenylmaleimide" Eur. J. Org. Chem. 2002, 947-964.
  52. K. Wojciechowski "1,3-Dihydro-2,1-benzisothiazole 2,2-Dioxides (Benzosultams) in Organic Synthesis" Heterocycles 2002, 57, 1717-1740 (Review).
  53. K. Wojciechowski, U. Siedlecka, H. Modrzejewska, S. Kosiński "Reactions of 6-(dichloromethylene)-cyclohexa-2,4-dien-1-alkylimines with amines" Tetrahedron 2002, 58, 7583-7588.
  54. K. Wojciechowski, H. Modrzejewska "Reactions of 1-arylbuta-1,3-dienes generated from 3-allyl-1,3-dihydro-benzisothiazole 2,2-dioxides" Pol. J. Chem. 2002, 76, 1587-1593.
  55. A. Chrostowska,  J.-M. Sotiropoulos, G. Pfister-Guillouzo, K. Wojciechowski "UV Photoelectron Spectroscopy Studies of the Diazaxylylenes Generated from Amino(hydroxymethyl)pyridines" Pol. J. Chem. 2003, 77, 535-545.
  56. K. Wojciechowski, H. Modrzejewska "Vicarious Nucleophilic Substitution of Hydrogen in Nitroarenes with Carbanions of in situ generated 1-Alkyl-3-chloro-1,3-dihydro-2,1-benzisothiazole 2,2-Dioxides" Synthesis 2003, 1503-1505.
  57. W. Danikiewicz, T. Bieńkowski, K. Wojciechowski "Application of electrospray ionization mass spectrometry for studies of anionic sigma-adducts of aromatic nitrocompounds" Tetrahedron Lett. 2004, 45, 931-934.
  58. M. Mąkosza, K. Wojciechowski "Nucleophilic Substitution of Hydrogen in Heterocyclic Chemistry" Chem. Rev. 2004, 104, 2631-2666 (Review)
  59. M. Mąkosza, K. Wojciechowski "Reactions of nucleophiles with nitroarenes: Efficient synthetic routes to indoles" in SELECTED METHODS FOR SYNTHESIS AND MODIFICATION OF HETEROCYCLES, vol. III (V.G. Kartsev Editor), IBS Press, Moscow 2004, 103-139 (Book chapter).
  60. K. Wojciechowski, K. Dolatowska "Generation of ortho-quinone methides upon thermal extrusion of sulfur dioxide from benzosultones" Tetrahedron 2005, 61, 8419-8422.
  61. H. Modrzejewska, K. Wojciechowski "Synthesis and reactions of 3-alkylsulfanyl-1,3-dihydro-2,1-benzisothiazole 2,2-dioxides" Tetrahedron 2005, 61, 8848-8854.
  62. R. Szmigielski, W. Danikiewicz, K. Dolatowska, K. Wojciechowski „Retro Diels-Alder and other electron ionization-induced fragmentation reactions of 1,2,3,4-tetrahydrobenzopyran-2,3-dicarboxylic acid derivatives” Int. J. Mass Spectrom. 2006, 248, 148-154.
  63. H. Modrzejewska, K. Wojciechowski " Reactions of aza-ortho-xylylenes generated from 3-aryl-2,1-benzisothiazoline 2,2-dioxides" Pol. J. Chem. 2006, 80, 1695-1702.
  64. H. Modrzejewska, K. Wojciechowski "Synthesis and Reactions of 3-Halogeno-3-methylbenzosultams" Pol. J. Chem. 2008, 82, 585-589.
  65. H. Modrzejewska, K. Wojciechowski "Generation of Arylcyclopenta-1,3-dienes from Cyclopenteno-spiro-benzosultams. Synthesis of 2-Arylnorbornenes" Synlett 2008, 2465-2470.
  66. Z. Wróbel, K. Wojciechowski, A. Kwast, N. Gajda "Short and Simple Method of Synthesis of Some Pyrrolo[3,2-b]quinoline Derivatives from Easily Available Nitrobenzene Derivatives" Synlett 2010, 2435-2438.
  67. M. Mąkosza, K. Wojciechowski "Nucleophilic Substitution of Hydrogen - An Efficient Tool in Synthesis of Heterocyclic Compounds " in Targets in Heterocyclic Systems. Chemistry and Properties. Vol 14. (O. A. Attanasi and D. Spinelli, Eds.) Societa Chimica Italiana, Roma 2011, 19-48 (Book Chapter).
  68. Z. Wróbel, K. Wojciechowski "Synthesis of Substituted 3-Cyano- and 3-(Arenesulfonyl)indoles from ortho-Nitrobenzyl Cyanides and Sulfones" Synlett 2011, 2567-2571.
  69. R. Bujok, Z. Wróbel, K. Wojciechowski "Expedient Synthesis of 1-Hydroxy-4- and 1-Hydroxy-6-nitroindoles” Synlett 2012, 1315-1320.
  70. R. Bujok, A. Trawczyński, Z. Wróbel, K. Wojciechowski "New Simple Synthesis of Quinoline-4-carbonitriles" Synlett 2012, 2682-2685.
  71. A. Trawczyński, R. Bujok, Z. Wróbel, K. Wojciechowski "Simple synthesis of pyrrolo[3,2-e]indole-1-carbonitriles" Beilstein J. Org. Chem. 2013, 9, 934–941. (PDF, HTML)
  72. Z. Wróbel, M. Więcław, R. Bujok, K. Wojciechowski "Synthesis of pyrrolo[3,2-a]phenazines from 5-nitroindoles and anilines" Monatshefte Chem. 2013,  144, 1847-1853 (OPEN ACCESS)
  73. M. Mąkosza, K. Wojciechowski "Nucleophilic Substitution of Hydrogen in Arenes and Heteroarenes" Top. Heterocycl. Chem. 2014, 37, 51-106 (Review).
  74. M. Mąkosza, K. Wojciechowski "Synthesis of Heterocycles via Nucleophilic Substitution of Hydrogen in Nitroarenes" Heterocycles 2014, 88, 75-101 (Review).
  75. M. Mąkosza, K. Wojciechowski "Application of Nucleophilic Substitution of Hydrogen in Nitroarenes to the Chemistry of Indoles" Chem. Heterocycl. Comp. 2015, 51, 210-222 (Review).
  76. K. Anczkiewicz, M. Królikiewicz, Z. Wróbel, K. Wojciechowski "Synthesis of 4-(4-toluenesulfonyl)quinolines from nitroarenes and allyl sulfones using step-by-step procedure" Tetrahedron 2015, 71 (23), 3924-3931. (PDF, HTML)
  77. M.Więcław, M. Bobin, A. Kwast, R. Bujok, Z. Wróbel, K. Wojciechowski "General synthesis of 2,1-benzisoxazoles (anthranils) from nitroarenes and benzylic C-H acids in aprotic media promoted by combination of strong bases and silylating agents" Mol. Divers. 2015, 19 (4), 807-816. (OPEN ACCESS)
  78. M. Nowacki, K. Wojciechowski "Simple synthesis 11-substituted norcryptotackieine derivatives" RSC Adv. 2015, 5, 94296-94303.
  79. R. Bujok, Z. Wróbel, K. Wojciechowski "Simple synthesis of 4-cyanoquinoline N-oxides" Tetrahedron Lett. 2016, 57 (9), 1014-1018.
  80. M. Nowacki, K. Wojciechowski "Transition-Metal-Free Direct Synthesis of Tetra- and Pentacyclic Azaheteroarenes via [3+3] Annulation of Nitroarenes and Benzyl-Type Carbanions Mediated by Silylating Agents" ChemistrySelect 2016, 1 (15), 4886–4890.
  81. R. Bujok, P. Cmoch, Z. Wróbel, K. Wojciechowski „Transition-metal-free synthesis of 3-(1-pyrrolidinyl)-quinolines and 3-(1-pyrrolidinyl)quinoline 1-oxides via a one-pot reaction of 3-(1-pyrrolidinyl)crotonates with nitrobenzenes” Org. Biomol. Chem. 2017, 15, 2397-2402 ( DOI: 10.1039/c6ob02658c) (OPEN ACCESS)
  82. M. Nowacki, K. Wojciechowski "Synthesis of [1]Benzothieno[2,3-b]quinolines via Transition-Metal-Free [3+3] Annulation of Nitroarenes and Benzo[b]thiophen-3-ylacetonitrile or 3-Phenylsulfonylmethyl)benzo[b]thiophene Carbanions" Synthesis 2017, 49 (16), 3794-3800. (DOI: 10.1055/s-0036-1588426)
  83. M. Nowacki, K. Wojciechowski "Transition-metal-free [3+3] annulation of indol-2-ylmethyl carbanions to nitroarenes. A novel synthesis of indolo[3,2-b]quinolines (quindolines)" Beilstein J. Org. Chem. 2018, 14, 194-202.  (DOI:10.3762/bjoc.14.14)   (OPEN ACCESS)
  84. M. Mąkosza, M. Bechcicka, K. Wojciechowski "Simple synthesis of dimethyl nitrobenzhydrylphosphonates and heteroarylnitroarylacetonitriles via VNS reaction" Synthesis 2020, in press.
    Last update 15.07.2020